Sign in
Back
A New Convenient Preparation of Thiol Esters Utilizing N-Acylbenzotriazoles
Journal article   Peer reviewed

A New Convenient Preparation of Thiol Esters Utilizing N-Acylbenzotriazoles

Alan R. Katritzky, Aleksandr A. Shestopalov and Kazuyuki Suzuki
Synthesis (Stuttgart), Vol.2004(11), pp.1806-1813
03/08/2004
DOI: https://doi.org/10.1055/s-2004-829126

Abstract

paper
ABSTRACT Diverse thiol esters were synthesized in good to excellent yields (76-99%) by reactions of thiophenol, benzyl mercaptan, ethyl­ mercaptoacetate, and mercaptoacetic acid with N-acylbenzo­triazoles under mild conditions. These results demonstrate the utility of N-acylbenzotriazoles as mild S-acylating agents, especially when the corresponding acid chlorides are not readily available.

Metrics

1 Record Views

Details