A facile route to 2-substituted N-Boc pyrrolidines

Alan R Katritzky; Zhushou Luo; Yunfeng Fang

doi:10.1016/S0040-4039(00)01763-9

Back

A facile route to 2-substituted N-Boc pyrrolidines

Journal article

Peer reviewed

A facile route to 2-substituted N-Boc pyrrolidines

Alan R Katritzky, Zhushou Luo and Yunfeng Fang

Tetrahedron letters, Vol.41(49), pp.9691-9693

02/12/2000

DOI: https://doi.org/10.1016/S0040-4039(00)01763-9

Abstract

dipole stabilization

intramolecular cyclization

pyrrolidine

Dipole stabilized carbanion 2 cyclizes to afford the key intermediate 2-benzotriazolyl- N-Boc-pyrrolidine 3, which undergoes nucleophilic displacement of the benzotriazolyl group to afford various 2-substituted- N-Boc-pyrrolidines in good yields.

Metrics

1 Record Views

Details

Title: A facile route to 2-substituted N-Boc pyrrolidines
Creators - without role: Alan R Katritzky - University of Florida
Zhushou Luo - University of Florida
Yunfeng Fang - University of Florida
Publication Details: Tetrahedron letters, Vol.41(49), pp.9691-9693
Publisher: Elsevier Ltd
Identifiers: 9935625108331
Academic Unit: King Abdulaziz University
Language: English
Resource Type: Journal article