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Addressing the metabolic activation potential of new leads in drug discovery: a case study using ion trap mass spectrometry and tritium labeling techniques
Journal article   Peer reviewed

Addressing the metabolic activation potential of new leads in drug discovery: a case study using ion trap mass spectrometry and tritium labeling techniques

Koppara Samuel, Wenji Yin, Ralph A. Stearns, Yui S. Tang, Ashok G. Chaudhary, James P. Jewell, Thomas Lanza Jr, Linus S. Lin, William K. Hagmann, David C. Evans, …
Journal of mass spectrometry, Vol.38(2), pp.211-221
02/2003
PMID: 12577288

Abstract

bioactivation covalent binding glutathione conjugates ion trap mass spectrometry microsomes reactive metabolites tritium labeling

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