Efficient N-Aroylation of Substituted Indoles with N-Aroylbenzotriazoles

Alan R. Katritzky; Levan Khelashvili; Prabhu P. Mohapatra; Peter J. Steel

doi:10.1055/s-2007-990889

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Efficient N-Aroylation of Substituted Indoles with N-Aroylbenzotriazoles

Journal article

Peer reviewed

Efficient N-Aroylation of Substituted Indoles with N-Aroylbenzotriazoles

Alan R. Katritzky, Levan Khelashvili, Prabhu P. Mohapatra and Peter J. Steel

Synthesis (Stuttgart), Vol.2007(23), pp.3673-3677

03/12/2007

DOI: https://doi.org/10.1055/s-2007-990889

Abstract

paper

Abstract Stable and easily accessible N-aroylbenzotriazoles react with indoles in the presence of a base to afford the corresponding N-aroylindoles in yields averaging 70%. This method is effective even when both coupling reagents possess electron-donating substituents.

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Title: Efficient N-Aroylation of Substituted Indoles with N-Aroylbenzotriazoles
Creators - without role: Alan R. Katritzky - Center for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA
Levan Khelashvili - Center for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA
Prabhu P. Mohapatra - Center for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, FL 32611-7200, USA
Peter J. Steel - University of Canterbury
Publication Details: Synthesis (Stuttgart), Vol.2007(23), pp.3673-3677
Identifiers: 9935806608331
Academic Unit: King Abdulaziz University
Language: English
Resource Type: Journal article