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FACILE SYNTHESIS OF beta-LACTAM-GRAFTED SPIROOXINDOLOPYRROLIDINE THROUGH REGIOSELECTIVE 1,3-DIPOLAR CYCLOADDITION REACTION
Journal article   Peer reviewed

FACILE SYNTHESIS OF beta-LACTAM-GRAFTED SPIROOXINDOLOPYRROLIDINE THROUGH REGIOSELECTIVE 1,3-DIPOLAR CYCLOADDITION REACTION

Natarajan Arumugam and Raghavachary Raghunathan
Synthetic communications, Vol.41(18), pp.2747-2755
15/09/2011

Abstract

Chemistry Chemistry, Organic Physical Sciences Science & Technology
One-pot synthesis of novel beta-lactam-grafted spiropyrrolidines has been accomplished in good yield via a facile [3+2] cycloaddition reaction of azomethine ylides, derived from beta-lactam aldehyde and sarcosine, with various p-substituted (E)-2-oxoindoline-3-ylidene acetophenone derivatives as dipolarophiles. The reaction gave excellent yields of the products when carried out under microwave irradiation.

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