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Ligation of anti-cancer drugs to self-assembling ultrashort peptides by click chemistry for localized therapy
Journal article   Peer reviewed

Ligation of anti-cancer drugs to self-assembling ultrashort peptides by click chemistry for localized therapy

Michael R. Reithofer, Kiat-Hwa Chan, Anupama Lakshmanan, Dang Hoang Lam, Archana Mishra, Began Gopalan, Mangesh Joshi, Shu Wang and Charlotte A. E. Hauser
Chemical science (Cambridge), Vol.5(2), pp.625-630
01/01/2014

Abstract

Chemistry Chemistry, Multidisciplinary Physical Sciences Science & Technology
Self-assembling ultrashort peptides from aliphatic amino acids were functionalized with platinum anticancer drugs by click chemistry. Oxaliplatin-derived hybrid peptide hydrogels with up to 40% drug loading were tested for localized breast cancer therapy. Stably injected gels showed significant tumor growth inhibition in mice and a better tolerance compared to the free platinum drug.

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