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Synthesis of thiazolyl and thieno cholestane derivatives: a novel class of potent antiinflammatory steroids
Journal article   Peer reviewed

Synthesis of thiazolyl and thieno cholestane derivatives: a novel class of potent antiinflammatory steroids

G A Elmegeed, W W Wardakhan and A R Baiuomy
Pharmazie, Vol.60(5), pp.328-333
05/2005
PMID: 15918579

Abstract

Animals Anti-Inflammatory Agents - chemical synthesis Anti-Inflammatory Agents - pharmacology Carrageenan Cholestanes - chemical synthesis Cholestanes - pharmacology Edema - chemically induced Edema - prevention & control Heterocyclic Compounds - chemical synthesis Heterocyclic Compounds - pharmacology Indicators and Reagents Magnetic Resonance Spectroscopy Male Rats Rats, Sprague-Dawley
The reactivity of 5alpha-cholestan-3-one (1) towards the formation of thiazolyl derivatives of potential antiinflammatory activity was studied. Also starting with the aminothieno[2',3': 2,3]cholestane derivative 8 several thiazolylthieno[2',3':2,3]cholestane derivatives were synthesized. The structures of the new compounds were established based on the analytical and spectral data and the in vivo antiinflammatory activities of some of these compounds were investigated.

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